Zu "409351-28-6" wurden 2 Artikel gefunden!
Für die Filterung wurden keine Ergebnisse gefunden!
VU0152100
Artikelnummer: TGM-T17238-100mg
Description: VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM). Target: AChR. Smiles: COc1ccc(CNC(=O)c2sc3nc(C)cc(C)c3c2N)cc1. References: Brady AE, et al. Centrally active allosteric potentiators of the M4 muscarinic acetylcholine receptor reverse amphetamine-induced...
| Schlagworte: | VU152100 |
| Anwendung: | Muscarinic M4 receptor positive allosteric modulator |
| CAS | 409351-28-6 |
| MW: | 341.43 D |
ab 34,00 €
VU0152100
Artikelnummer: Cay32968-10
VU0152100 is a positive allosteric modulator of M4 muscarinic acetylcholine receptors. It potentiates calcium mobilization induced by acetylcholine (ACh) in CHO-K1 cells expressing the rat M4 receptor with an EC50 value of 380 nM. VU0152100 is selective for M4 over M1, M2, M3 and M5 receptors, as well as a panel of...
| Schlagworte: | 3-amino-N-[(4-methoxyphenyl)methyl]-4,6-dimethyl-thieno[2,3-b]pyridine-2-carboxamide |
| Anwendung: | Muscarinic M4 receptor positive allosteric modulator |
| CAS | 409351-28-6 |
| MW: | 341.4 D |
ab 126,00 €
