Zu "401907-26-4" wurden 2 Artikel gefunden!

Für die Filterung wurden keine Ergebnisse gefunden!
JYL 1421
JYL 1421

Artikelnummer: TGM-T15634-100mg

Description: JYL 1421 (SC 0030) is an antagonist of TRPV1 receptor (IC50 = 8 nM). Target: TRP/TRPV Channel. Smiles: CC(C)(C)c1ccc(CNC(=S)NCc2ccc(NS(C)(=O)=O)c(F)c2)cc1. References: Jakab B, et al. Pharmacological characterization of the TRPV1 receptor antagonist JYL1421 (SC0030) in vitro and in vivo in the rat. Eur...
Schlagworte: SC 0030
Anwendung: Selective TRPV1 receptor antagonist
CAS 401907-26-4
MW: 423.57 D
ab 751,00 €
Bewerten
JYL1421
JYL1421

Artikelnummer: Cay20458-500

JYL1421 is an antagonist of transient receptor potential vanilloid 1 (TRPV1). It inhibits calcium uptake induced by capsaicin (Cay-92350, Cay-10010743) in CHO cells expressing rat TRPV1 (EC50 = 9.2 nM). JYL1421 inhibits capsaicin-induced release of the neuropeptides somatostatin, substance P (Cay-24035), and...
Schlagworte: N-[4-[[[[[[4-(1,1-dimethylethyl)phenyl]methyl]amino]thioxomethyl]amino]methyl]-2-fluorophenyl]-methanesulfonamide
Anwendung: Selective TRPV1 receptor antagonist
CAS 401907-26-4
MW: 423.6 D
ab 66,00 €
Bewerten