Zu "2062-78-4" wurden 2 Artikel gefunden!
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Pimozide
Artikelnummer: Cay16222-50
Pimozide is a dopamine receptor antagonist (Kis = 2.4, 0.3, and 1.8 nM for D2, D3, and D4 receptors, respectively). It also binds to eight additional receptors (Kds = 25-3,100 nM for the human receptors) and inhibits the voltage-gated sodium channel Nav1.2 and the voltage-gated potassium channel Kv11.1 (IC50s = 42...
| Schlagworte: | NSC 170984, R 6238, 1-[1-[4,4-bis(4-fluorophenyl)butyl]-4-piperidinyl]-1,3-dihydro-2H-benzimidazol-2-one |
| Anwendung: | Dopamine D2/D3-receptor antagonist |
| CAS | 2062-78-4 |
| MW: | 461.6 D |
ab 44,00 €
Pimozide
Artikelnummer: TGM-T2546-1mL
Description: Pimozide (R6238) is a diphenylbutylpiperidine derivative and a dopamine antagonist with the antipsychotic property. Pimozide selectively inhibits type 2 dopaminergic receptors in the central nervous system (CNS), thereby decreasing dopamine neurotransmission and reducing the occurrence of the motor and...
| Schlagworte: | R6238 |
| Anwendung: | Targets dopamine receptor D2 (DRD2) |
| CAS | 2062-78-4 |
| MW: | 461.55 D |
ab 31,00 €
