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Perlapine
Perlapine

Artikelnummer: TGM-T33937-10mg

Description: Perlapine is an effective and selective HM3DQ DREADD agonist (EC50 = 2.8 nM). Target: Others. Smiles: N=1C=2C=CC=CC2CC=3C=CC=CC3C1N4CCN(C)CC4. References: Meltzer HY, Fessler RG, Fang VS. Perlapine: relationship between stimulation of prolactin secretion and antipsychotic activity. Psychopharmacology...
Anwendung: Melatonin receptor 1A/B agonist
CAS 1977-11-3
MW: 291.39 D
ab 142,00 €
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Perlapine
Perlapine

Artikelnummer: Cay17756-10

Perlapine is an atypical neuroleptic that blocks dopamine and serotonin (5-HT) receptors (Kis = 60, 30, and 30 nM for D2, D4, and 5-HT2A, respectively). Perlapine is also an agonist for hM3Dq, a designer receptor exclusively activated by designer drugs (DREADDs) derived from the human muscarinic acetylcholine M3...
Schlagworte: 6-(4-Methyl-1-piperazinyl)morphanthridine, NSC 291840, 6-(4-methyl-1-piperazinyl)-11H-dibenz[b,e]azepine
Anwendung: Melatonin receptor 1A/B agonist
CAS 1977-11-3
MW: 291.4 D
ab 78,00 €
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