Zu "183232-66-8" wurden 3 Artikel gefunden!
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AM251
Artikelnummer: Cay71670-10
AM251 is a cannabinoid 1 (CB1) receptor 1 antagonist. It binds to CB1 receptors in rat forebrain membrane preparations (Ki = 7.5 nM) and is selective over CB2 receptors in mouse spleen preparations (Ki = 2,290 nM) in radioligand binding assays. AM251 inhibits GTPgammaS binding induced by the CB receptor agonist CP...
| Schlagworte: | 1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide |
| Anwendung: | SR 141716A analog |
| CAS | 183232-66-8 |
| MW: | 555.2 D |
ab 67,00 €
AM251
Artikelnummer: TGM-T1915-100mg
Description: AM251 is a effective CB1 receptor antagonist (IC50/Ki: 8 /7.49 nM) that displays 306-fold selectivity over CB2 receptors, also effective GPR55 agonist (EC50: 39 nM). Target: Cannabinoid Receptor, GPR. Smiles: CC1=C(N(N=C1C(NN2CCCCC2)=O)C3=C(Cl)C=C(Cl)C=C3)C4=CC=C(I)C=C4. References: Liao C, et al....
| Anwendung: | SR 141716A analog |
| CAS | 183232-66-8 |
| MW: | 555.24 D |
ab 43,00 €
AM251
Artikelnummer: LKT-A480000.5
CB1 receptor antagonist/ inverse agonist.
| Schlagworte: | AM-251, AM 251, 1-(2,4-Dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide |
| Anwendung: | SR 141716A analog |
| CAS | 183232-66-8 |
| MW: | 555.24 D |
ab 110,00 €
