Zu "168482-23-3" wurden 2 Artikel gefunden!
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SHU 9119
Artikelnummer: TGM-T16879-1mg
Description: SHU 9119 is an effective human melanocortin 3 and 4 receptors (MC3/4R) antagonist and a partial MC5R agonist (IC50: 0.23, 0.06, and 0.09 nM for human MC3R, MC4R and MC5R, respectively). Target: Others. Smiles:...
| Anwendung: | MC1R agonist, MC4R antagonist |
| CAS | 168482-23-3 |
| MW: | 1074.258 D |
ab 189,00 €
SHU9119 (trifluoroacetate salt)
Artikelnummer: Cay24152-1
SHU9119 is an agonist of melanocortin receptor 1 (MC1R) and antagonist of MC4R (IC50s = 1.2 and 2.9 nM, respectively, for displacement of melanocortin). It induces cAMP formation in HEK293 cells expressing human MC1R (EC50 = 1.11 nM), but inhibits cAMP formation in cells expressing human MC4R. In rats, SHU9119 (24...
| Schlagworte: | N-acetyl-L-norleucyl-L-alpha-aspartyl-L-histidyl-3-(2-naphthalenyl)-D-alanyl-L-arginyl-L-tryptophyl-L-lysinamide,... |
| Anwendung: | MC1R agonist, MC4R antagonist |
| CAS | 168482-23-3 |
| MW: | 1074.2 D |
ab 104,00 €
