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MJN110
MJN110

Artikelnummer: TGM-T5815-100mg

Description: MJN110 (Cravatt Reagent) is a potent and selective MAGL inhibitor. Cravatt Reagent inhibits MAGL (IC50 = 9.1 nM). MJN110(Cravatt Reagent) Produces Opioid-Sparing Effects in a Mouse Neuropathic Pain Model. Target: Lipase. Smiles: Clc1ccc(cc1)C(N1CCN(CC1)C(=O)ON1C(=O)CCC1=O)c1ccc(Cl)cc1. References:...
Schlagworte: Cravatt Reagent
Anwendung: MGLL inhibitor
CAS 1438416-21-7
MW: 462.33 D
ab 43,00 €
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MJN110
MJN110

Artikelnummer: Cay17583-5

Endocannabinoids such as 2-arachidonoyl glycerol (2-AG, Cay-62160) and arachidonoyl ethanolamide (AEA, Cay-90050) are biologically active lipids that are involved in a number of synaptic processes including activation of cannabinoid receptors. Monoacylglycerol lipase (MAGL) is a serine hydrolase responsible for the...
Schlagworte: 2,5-Dioxopyrrolidin-1-yl 4-[bis(4-chlorophenyl)methyl]piperazine-1-carboxylate,...
Anwendung: MGLL inhibitor
CAS 1438416-21-7
MW: 462.3 D
ab 112,00 €
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