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BQ-123
Artikelnummer: TGM-T6792-100mg
Description: BQ-123 is a selective endothelin A receptor (ETA) antagonist with IC50 of 7.3 nM. Phase 2. Target: Endothelin Receptor. Smiles: [H][C@@]12CCCN1C(=O)[C@@]([H])(CC(O)=O)NC(=O)[C@@H](Cc1c[nH]c3ccccc13)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](NC2=O)C(C)C. References: Ihara M, et al. J Cardiovasc Pharmacol. 1992, 12,...
| Schlagworte: | BQ123 |
| Anwendung: | Endothelin receptor A antagonist |
| CAS | 136553-81-6 |
| MW: | 610.7 D |
ab 81,00 €
BQ-123 sodium salt
Artikelnummer: AG-CP3-0001-M001
Potent and selective endothelin receptor A (ETA) antagonist, suppresses the ET-1-induced decrease of LPL activity, shows protective effects in ischemic acute renal failure, neuroprotective, anti-hypertensive, inhibits ET-1 receptor binding and blocks Ca2 mobilization, cellular contraction and MAP kinase activation,...
| Schlagworte: | Endothelin Receptor A Antagonist BQ-123, cyclo(-D-Trp-D-Asp-Pro-D-Val-Leu) Na |
| Anwendung: | Endothelin receptor A antagonist |
| CAS | 136553-81-6 |
| MW: | 609,7 D |
ab 116,00 €
BQ-123
Artikelnummer: Cay19153-1
BQ-123 is a peptide endothelin type A (ETA) receptor antagonist (IC50 = 7.3 nM). It is selective for ETA over ETB receptors (Kis = 0.025 and 31 µM, respectively). BQ-123 inhibits growth of human pulmonary artery smooth muscle cells induced by endothelin-1 (ET-1, Cay-24127). It reverses ET-1-induced increases in mean...
| Schlagworte: | Cyclo(D-Trp-D-Asp-Pro-D-Val-Leu), cyclo(D-alpha-aspartyl-L-prolyl-D-valyl-L-leucyl-D-tryptophyl) |
| Anwendung: | Peptide ETA receptor antagonist |
| CAS | 136553-81-6 |
| MW: | 610.7 D |
ab 145,00 €
