Zu "121917-57-5" wurden 2 Artikel gefunden!
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(-)-Dizocilpine maleate
Artikelnummer: TGM-T6352-100mg
Description: (-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective, and non-competitive NMDA receptor antagonist, with a Kd of 37.2 nM in rat brain membranes. Target: NMDAR, iGluR. Smiles: OC(=O)\C=C/C(O)=O.C[C@@]12N[C@@H](Cc3ccccc13)c1ccccc21. References: Wong EH, et al. Proc Natl Acad Sci U S A,...
| Schlagworte: | (-)-MK 801 (Maleate), C13737, (-)-MK 801 Maleate |
| Anwendung: | NMDA receptor antagonist |
| CAS | 121917-57-5 |
| MW: | 337.37 D |
ab 45,00 €
(-)-MK-801 (maleate)
Artikelnummer: Cay27213-10
(-)-MK-801 is an NMDA receptor antagonist (Ki = 43 nM for inhibition of spermine binding) and an isomer of (+)-MK-801 (Cay-10009019). In vivo, (-)-MK-801 blocks generalized seizures in a mouse model of epilepsy (ED50 = 0.85 mg/kg) and increases horizontal locomotor activity in mice (ED50 = 2.71 mg/kg). (-)-MK-801...
| Schlagworte: | (5R,10S)-10,11-dihydro-5-methyl-5H-dibenzo[a,d]cyclohepten-5,10-imine, (2Z)-2-butenedioate |
| Anwendung: | NMDA receptor antagonist |
| CAS | 121917-57-5 |
| MW: | 337.4 D |
ab 44,00 €
