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Nav1.7 Blocker 52
Nav1.7 Blocker 52

Artikelnummer: Cay34477-5

Nav1.7 blocker 52 is an inhibitor of voltage-gated sodium channel 1.7 (Nav1.7, IC50 = 0.17 µM). It is selective for Nav1.7 over human-ether-a-go-go (hERG), also known as Kv11.1, Nav1.5, and Nav1.8 (IC50s = >10, 1.1, and 2.2 µM, respectively) but does inhibit Nav1.3 and Nav1.4 (IC50s = 0.3 and 0.4 µM, respectively)....
Schlagworte: TC-N 1752, Voltage-gated Sodium Channel 1.7,...
Anwendung: Nav1.7 inhibitor
CAS 1211866-85-1
MW: 516.5 D
ab 163,00 €
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