Zu "102394-31-0" wurden 2 Artikel gefunden!
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Otenzepad
Artikelnummer: TGM-T16411-100mg
Description: Otenzepad (AF-DX 116) is a selective M2 mAChR antagonist with IC50 values of 386 nM in rat heart and 640 nM in rabbit peripheral lung. Target: AChR. Smiles: CCN(CC)CC1CCCCN1CC(=O)N1c2ccccc2C(=O)Nc2cccnc12. References: Packard MG, et al. Post-training injection of the acetylcholine M2 receptor antagonist...
| Schlagworte: | AF-DX 116 |
| Anwendung: | Muscarinic acetylcholine receptor M2 antagonist |
| CAS | 102394-31-0 |
| MW: | 421.54 D |
ab 39,00 €
AF-DX 116
Artikelnummer: Cay30871-1
AF-DX 116 is an antagonist of M2 muscarinic acetylcholine receptors (Ki = 0.2 µM). It is selective for cardiac M2 over salivary gland M3 receptors (Ki = 5.01 µM) but also binds sympathetic ganglia M1 receptors (Ki = 0.81 µM). AF-DX 116 (0.1 µM) increases vagus nerve stimulation-induced increases in perfusion...
| Schlagworte: | 11-[2-[2-[(diethylamino)methyl]-1-piperidinyl]acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one |
| Anwendung: | Muscarinic acetylcholine receptor M2 antagonist |
| CAS | 102394-31-0 |
| MW: | 421.5 D |
ab 46,00 €
