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CRA-026440 hydrochloride
Artikelnummer: TGM-T10883L-5mg
Description: CRA-026440 hydrochloride is a potent and broad-spectrum HDAC inhibitor. CRA-026440 hydrochloride exhibits Ki values against recombinant HDAC isoenzymes HDAC1, HDAC2, HDAC3, HDAC6, HDAC8, and HDAC10 are 4 nM, 14 nM, 11 nM, 15 nM, 7 nM, and 20 nM, respectively. CRA-026440 hydrochloride exhibits antitumor...
| Schlagworte: | CRA-026440 hydrochloride(847460-34-8 Free base) |
| CAS | 847459-98-7 |
| MW: | 456.92 D |
ab 40,00 €
CSRM617 hydrochloride
Artikelnummer: TGM-T10896L-50mg
Description: CSRM617 hydrochloride is a selective small-molecule inhibitor of the transcription factor ONECUT2 (OC2, a master regulator of androgen receptor), with a Kd of 7.43 µM in SPR assays, directly binding to the OC2-HOX domain. CSRM617 hydrochloride induces apoptosis through the appearance of cleaved...
| Schlagworte: | CSRM617 hydrochloride(787504-88-5 Free base) |
| CAS | 1353749-74-2 |
| MW: | 291.69 D |
ab 54,00 €
AKT Kinase Inhibitor HCl
Artikelnummer: TGM-T10276L-5mg
Description: AKT Kinase Inhibitor HCl is an Akt inhibitor with antitumor activity. Target: Akt. Smiles: OCC#CC1=C(N=C(N2CC)C3=NON=C3N)C2=C(OCCCN)C=N1.Cl. References: Saverio Alberti, et al. Use of trop-2 as predictive marker of response to anti-tumor therapy based on inhibitors of cd9, akt and molecules of the...
| Schlagworte: | AKT Kinase Inhibitor HCl(842148-40-7 Free base) |
| MW: | 393.83 D |
ab 139,00 €
BMT-124110 Formate
Artikelnummer: TGM-T10572L-5mg
Description: BMT-124110 Formate is a selective AAK1 inhibitor (IC50: 0.9 nM) with anti-injury sensory activity.BMT-124110 Formate inhibits the BMP-2-inducible protein kinase BIKE with an IC50: 17 nM.BMT-124110 Formate inhibits the cell-cycle protein G-related BMT-124110 Formate inhibits the cell cycle protein...
| Schlagworte: | BMT-124110 Formate(1679371-59-5 Free base) |
| MW: | 344.41 D |
ab 194,00 €
A-317491 sodium salt hydrate
Artikelnummer: TGM-T10204-50mg
Description: A-317491 sodium salt hydrate is a non-nucleotide P2X3 and P2X2/3 receptor antagonist that inhibits receptor-mediated calcium flux. Target: Others. Smiles: O=C(O)C1=CC(C(N([C@H]2CCCC3=C2C=CC=C3)CC4=CC=CC(OC5=CC=CC=C5)=C4)=O)=C(C=C1C(O)=O)C(O)=O.[Na+].O. References: Hansen RR, Nasser A, Falk S, et al....
| Schlagworte: | A-317491 sodium salt hydrate (475205-49-3 free base) |
| MW: | 606.57 D |
ab 86,00 €
Apidaecin IB acetate
Artikelnummer: TGM-T10347L-10mg
Description: Apidaecin IB acetate is an insect antibacterial peptide. The minimum concentration of apidaecin IB acetate against Escherichia coli (E. coli ML35, o18k1h7 and ATCC 25922) is 8 µM. Target: Others. Smiles:...
| Schlagworte: | Apidaecin IB acetate (123276-94-8 Free base) |
| MW: | 2168.46 D |
ab 112,00 €
Arg-Gly-Asp-Ser acetate
Artikelnummer: TGM-T10366L-50mg
Description: Arg-Gly-Asp-Ser acetate is an integrin binding sequence that directly and specifically bind pro-caspase-8, pro-caspase-9 and pro-caspase-3, while it does not bind pro-caspase-1. Arg-Gly-Asp-Ser acetate inhibits integrin receptor function. Target: Integrin. Smiles:...
| Schlagworte: | Arg-Gly-Asp-Ser acetate(91037-65-9 free base) |
| MW: | 493.47 D |
ab 37,00 €
ATB107 hydrochloride
Artikelnummer: TGM-T10394L-10mg
Description: ATB107 hydrochloride is a novel and potent inhibitor of indole-3-glycerol phosphate synthase (IGPS) with a KD of 3 µM. Target: Others. Smiles: N1(C2=NC(NC3=CC=CC=C3)=NC(N/N=C4CN5CCC\4CC5)=N2)CCCCC1.Cl. References: Shen H, et al. A novel inhibitor of indole-3-glycerol phosphate synthase with activity...
| Schlagworte: | ATB107 hydrochloride(455325-51-6 Free base) |
| MW: | 428.96 D |
ab 60,00 €
Shepherdin 79-87 acetate
Artikelnummer: TGM-T12896L-10mg
Description: Shepherdin 79-87 acetate is a peptidomimetic antagonist of the complex between Hsp90 and survivin, another key regulator of tumor cell viability. Target: Survivin, HSP. Smiles:...
| Schlagworte: | Shepherdin 79-87 acetate (861224-28-4 free base) |
| MW: | 1009.14 D |
ab 147,00 €
WAY-213613 hydrochloride
Artikelnummer: TGM-T13330-10mg
Description: WAY-213613 hydrochloride is a potent, selective nonsubstrate reuptake inhibitor of GLT-1/EAAT2 with IC 50 of 85 nM. WAY-213613 hydrochloride inhibits EAAT1 and EAAT3 with IC50 values of 5 and 3.8 microM, respectively. WAY-213613 hydrochloride shows no activity at ionotropic and metabotropic glutamate...
| Schlagworte: | WAY-213613 hydrochloride (868359-05-1 free base) |
| CAS | 2450268-84-3 |
| MW: | 451.65 D |
ab 33,00 €
OTS186935 FA
Artikelnummer: TGM-T12344L1-10mg
Description: OTS186935 FA is a protein methyltransferase SUV39H2 inhibitor.OTS186935 FA inhibits tumor growth in MDA-MB-231 breast cancer cells and A549 lung cancer cells. Target: Histone Methyltransferase. Smiles: COC1=C(C2=CN(C=CC(N3C[C@H](CC3)NCC4=CC=NC=C4)=C5)C5=N2)C=C(C(OC)=C1)Cl.[H]C(O)=O. References:...
| Schlagworte: | OTS186935 FA(2093400-18-9 Free base) |
| MW: | 509.98 D |
ab 98,00 €
Theodrenaline hydrochloride
Artikelnummer: TGM-T13142L-5mg
Description: Theodrenaline hydrochloride is an inhibitor targeting SARS-CoV-2 for the study of hypotension induced by spinal anesthesia. Target: SARS-CoV. Smiles: O=C1C2=C(N(C)C(N1C)=O)N=CN2CCNCC(C3=CC=C(C(O)=C3)O)O.Cl. References: Kloth B, et al. AkrinorTM, a Cafedrine/ Theodrenaline Mixture (20:1), Increases Force...
| Schlagworte: | Theodrenaline hydrochloride(13460-98-5 Free base) |
| CAS | 2572-61-4 |
| MW: | 411.84 D |
ab 158,00 €