UR-144 N-(5-chloropentyl) analog

UR-144 (Cay-11502) is a potent synthetic cannabinoid (CB) which preferentially binds the peripheral CB2 receptor (Ki = 1.8 nM) over the central CB1 receptor (Ki = 150 nM). UR-144 N-(5-chloropentyl) analog differs from UR-144 by having a chlorine atom on the terminal carbon of the alkyl group. The biological activities of this compound have not been characterized. This product is intended for forensic and research applications.Formal Name: (1-(5-chloropentyl)-1H-indol-3-yl)(2,2,3,3-tetramethylcyclopropyl)methanone. CAS Number: 1445577-42-3. Molecular Formula: C21H28ClNO. Formula Weight: 345.9. Purity: >98%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF: 14 mg/ml, DMF:PBS(pH7.2) (1:2): 0.3 mg/ml, DMSO: 5 mg/ml, Ethanol: 5 mg/ml. lambdamax: 218, 246, 304 nm. SMILES: O=C(C1C(C)(C)C1(C)C)C2=CN(CCCCCCl)C3=C2C=CC=C3. InChi Code: InChI=1S/C21H28ClNO/c1-20(2)19(21(20,3)4)18(24)16-14-23(13-9-5-8-12-22)17-11-7-6-10-15(16)17/h6-7,10-11,14,19H,5,8-9,12-13H2,1-4H3. InChi Key: CKIOITGXSRFWIS-UHFFFAOYSA-N.