N-(p-amylcinnamoyl) Anthranilic Acid

N-(p-amylcinnamoyl) Anthranilic acid (ACA) is a channel blocker that acts on several transient receptor potential (TRP) channels, including TRPM2, TRPM8, and TRPC6 (IC50 = 1.7, 3.8, and 2.3 µM, respectively). It is a weak inhibitor of TRPV1. ACA is also an inhibitor of phospholipase A2, blocking the release of arachidonic acid when given at 50 µM.Formal Name: 2-[[1-oxo-3-(4-pentylphenyl)-2-propen-1-yl]amino]-benzoic acid. CAS Number: 110683-10-8. Synonyms: ACA. Molecular Formula: C21H23NO3. Formula Weight: 337.4. Purity: >95%. Formulation: (Request formulation change), A crystalline solid. Solubility: DMF: 5 mg/ml, DMSO: 11.1 mg/ml, DMSO:PBS (pH 7.2) (1:1): 0.5 mg/ml, Ethanol: 5 mg/ml. lambdamax: 216, 300, 323 nm. SMILES: CCCCCC1=CC=C(/C=C/C(NC2=CC=CC=C2C(O)=O)=O)C=C1. InChi Code: InChI=1S/C21H23NO3/c1-2-3-4-7-16-10-12-17(13-11-16)14-15-20(23)22-19-9-6-5-8-18(19)21(24)25/h5-6,8-15H,2-4,7H2,1H3,(H,22,23)(H,24,25)/b15-14+. InChi Key: GAMRBCZMOOMBSQ-CCEZHUSRSA-N.